Ko te tarukino "Ksarelto" tohutohu mō te whakamahi rite te tikanga ki te tohu, ko te anticoagulant o mahi tika. I roto i te pūtake o tenei tarukino ko te inhibition tika o te tauwehe Xa. I tua atu, kua he selectivity āhua tiketike tenei tarukino. Ka rite ki hoki ona pharmacokinetics, Kei te tino tere whenumi reira, pa kukū mōrahi i roto i te toto i muri i rua anake ki wha haora i muri i whakahaere-waha. Ki te kōrero tatou e pā ana ki te āhuatanga o te excretion tiketike o te tarukino, me te mimi me feces whakaaturia e pā ana ki 92-95% o te rongoā "Ksarelto". Tohutohu mō te whakamahi (utu, i te ara, tenei te tikanga ko e pā ana ki 1500 moni) tuhia konei e rau te toe wahi te tinana i roto i te puka taui i te excretion tākihi.
Wātea tenei anticoagulant i te puka o papa a tawhio māwhero pouri te tae whero-parauri ranei, kei roto i roto i tona hanganga tekau, rima e rua tekau ranei milligrams o rivaroxaban micronized. Ngaahi houalotú he matū pērā i croscarmellose konutai, te konutai lauryl pūkawa, hypromellose 5cP, microcrystalline cellulose, stearate konupora me te monohydrate reihuka. Ko te hanganga anga ngā Titanium hāorarua, Macrogol 3350 me te whero waikura ferric. I tua atu, kei te rōrahi iti hypromellose 5cP.
Whakaritea pire "Ksarelto" tohutohu mō te whakamahi tikanga tūtohutia hoki tūroro hunga i pehia mua ngā tukanga hāparapara i runga i nga topito o raro. Hoki tenei kāwai o te iwi te mahi anticoagulant hei mehua ārai whai hua mo te whanaketanga o te thromboembolism venous heke mai. I tua atu, i te tarukino "Ksarelto" tino tika ana mō te ārai o te hohokitanga o DVT me PE. Hoki, kia whakamahia tenei taputapu mo te ārai o te patunga i roto i te iwi ki te fibrillation Atrial, momo kore-valvular. Kia kore ai te whanaketanga o te thromboembolism pūnahanaha me te maimoatanga o te Thrombosis rua hohonu me te occlusion whakapeka o te iatuku pūkahukahu taunaki tango hoki pire "Ksarelto" ako ā-ringa.
Whakamahia te tino tenei anticoagulant contraindicated hoki te iwi ki te gastrointestinal, intracranial ranei tetahi atu momo o toto, he ahua nui o hēnga o ōna whatukuhu ātete ranei ki galactose. I roto i te take ki te hypersensitivity o te manawanui rivaroxaban ranei tauhohenga pāwera ki ētahi atu excipients whakarārangitia i roto i te hanganga, me kore e tangohia e te tarukino "Ksarelto". Tohutohu mō te whakamahi opani whakarite ia kaha me te wā hapūtanga. E hoki Contraindications reihuka kātaki'i, maimoatanga ki ētahi atu anticoagulants, mate ate, haere tahi i te coagulopathy, me ngā āhuatanga e pā ana ki te mōrea tiketike o te toto nui. I tua atu, e kore koutou e taea e te tango i te wahine rongoā, te u, me tangata kahore i nei i tae te tau o waru.