Hauora, Mau faaineineraa
Drug "Sotageksal", analogs me urupare ki runga ki a ratou
Arrhythmia - Ko te momo o te auau ngakau, he rerekē i te manawataki pakohu noa nei. A, no te arrhythmias i roto i te tangata i reira he kotahi e rave rahi e aore maumaui o te ngakau. kia tapaea te māuiuitanga rite te auau me te mana amplification auau ngakau (tachycardia) me, hei kōrero, he hekenga i roto i to ratou (bradycardia). Taupatupatu ki te mahi o te uaua ngakau me kei roto i te tangata hauora. Heoi, i roto i te nuinga o te wā, ko te arrhythmia roto i te taha ki ētahi atu mate cardiac. Ko meá he āhua pērā i roto i taua i te nui haere excitability o kiko ngakau - myocardium, e taea arahi hopea ki te kore te ngakau, ki te mahue kore maimoatia.
i reira he ngaahi teuteu motuhake mo te māori o auau ngakau, tetahi o te mea "Sotageksal". Analogues o te tarukino te hoki whānui e whakamahia ana i roto i te mahi hauora. no enei taero ki te rōpū o ngā rongoā e whai mahi antiarrhythmic, me beta-blockers. A, no te ingested, te aukati ratou nga receptors beta-adrenergic, e kua kei roto i te uaua maeneene, uaua cardiac me ētahi atu te kopa, a he kawenga mō te whakautu a te tinana ki te pānga o te ahotea. kardioeffekt whānui ko ki te whakaiti i te auau me te kaha o te auau ngakau, heke cardiac kawenga. Ka rite ki te kitea ano i te pānga pūnahanaha e tukupu ana o te pēhanga toto i runga i te taiepa o nga oko coronary.
te raau taero
"Sotalol» (Sotalol) - ohi e te ingoa ao i roto i te ao o te tarukino "Sotageksal". kia whai Analogs o te hanganga i te pānga antiarrhythmic rerekē, engari rite. Ko te taonga kaha matua "Sotageksal" kei sotalol hydrochloride. I tua atu, ngā reira he maha iti o ngā wāhanga ngaahi houalotú. I roto ia ratou, - cellulose, monohydrate reihuka, te kānga māngaro, stearate konupora me te tahi atu uwhi.
Ko te ora papa o papa otinga injectable ranei he 5 tau.
"Sotageksal" analogues me Composition
Ko tētahi papa o tenei hua kei roto 40, 80 ranei 160 mg o taonga kaha. Kei te whakaputaina te reira i te nuinga rite papa a tawhio White ki tetahi taha paku ohu nei, me te whakairo ki te muru whakarāpopototanga. I runga i te hoki o te papa wahia e te tikanga o dosing mo te haratau o te tūponotanga. Kikī katoa i roto i te opupu o te 10 nga wahi, me pouaka pepa. kia ngā Ia paihere i te 1 ki te 10 opupu (o i te 10 ki te 100 nga wahi o papa).
Hoki, "Sotageksal" hua i roto i te puka o te otinga mō te werohia rō-uaua. Kei ia ampoule 4 ml o tarukino. I roto i te 1 ml o te otinga ko te 10 mg o taonga taketake parakore. kia tiakina te tarukino i te rā pouri me te wahi maroke, i roto i nei tamariki i he iti uru.
Analogs ki te taonga sotalol kaha e hangaia papa hydrochloride:
- "Sotaleks" (160 mg).
- "Soritmik" (e 0,16 g).
- "Sotalol Canon" (80 me 160 mg).
- "Darob" (80 me 160 mg).
- "Tenzol" (80 me 160 mg).
pānga pharmacological
"Sotageksal" analogues me taurite o te tarukino i te pānga anti-arrhythmic korerotia. tutuki ana tēnei e te viivii ore o to ratou kaha ki te ārai receptors β-adrenergic me tautāwhi i takere pāhare pāporo. whakanui i taero i te roanga o te ngātere me pūpū wā atria me ventricles. Whakanuia te reo o te uaua maeneene arahau me te kahu uaua o te taiepa oko. Whakaititia contractility myocardial.
hydrochloride Sotalol he huinga katoa o ngā āhuatanga. Kua he chronotropic kino, dromotropic, batmotroponoe me te pānga inotropic o te tarukino German "Sotageksal". Analogs, te hanganga o nei he ōrite, kia whai tetahi ingoa waitohu. E taea e ki te whakaiti i auau ngakau me o ratou kaha hoki ratou. No te mea o tenei hiahia mō te kohi hāora myocardial te nui iti. A, ka rite ki te hua, heke te kawenga i runga i te ngakau te.
Absorption me excretion o taero
he tere Drug absorption. Ko tōna bioavailability ko 90%, me te absorption - e pā ana ki 80%. I roto i 2.5-4 haora o kukū mōrahi o whakauru kaha tutuki te i muri i te fariiraa i te wē. I muri i whakahaere rō-uaua, he kitea i muri i 5-10 meneti kua te pānga. puta absorption i 20% pai me tere ki te tango koe i te rongoā i runga i te puku kau. Nā ki te meka e te memehatanga o te taonga i roto i te ngako te mea tino iti, kia kore sotalol hydrochloride e tangohia tukutahi ki ngā hua miraka me te ngako o te take kararehe.
Te kore he mea here ki pūmua toto, tohaina te raau taero i roto i te kopa me okana piringa whakanoho i roto i 3-4 ra o whakauru auau. I te wa ano, ka tutuki ana e ia he pānga pai i runga i takawhita. I roto i te inu cerebrospinal kore te mea neke atu i te 20% te kukū tarukino. Mahi i muri i werohia tonu ki runga ki te 2 haora. pānga tonu i muri i dosing waha o papa "Sotageksal" ki 12 haora. Analogs o te raau taero i roto i te hanganga i kei roto sotalol hydrochloride, e kore ano i haria ki te pākia e te whatukuhu, me excreted i roto i te mimi (90%) me te feces i toharite i roto i 10-20 haora.
Ko te aha tūroro ki te pūnaha tākihi me te mimi waimaero whakaatu te rongoā ki te inenga iti. Kei te maha iwi pakeke kitea ino e pā ana-tau o te mahi tākihi. whai wāhi ana tēnei ki te meka i whakaaturia te taonga kei te i te tere pōturi a kia kohikohi i roto i te tinana. Na reira, kia whakamahia tenei rōpū o tūroro te tarukino ki tūpato, me te takoto te inenga te takitahi.
tauturu te rongoa ki te haerenga i te utu o te hāora i roto i te kopa, faaore irritability, manukanuka, ahotea me ētahi atu āhuatanga e pā te auau me te kaha o contractions o te ngakau.
"Sotageksal": tohutohu mō te whakamahi
Kei te whakamahia Analogs o te tarukino me te kaihoko ki te ingoa taketake mō arrhythmias cardiac symptomatic, mo te maimoatanga o te ventricular arrythmia. Ko reira te mea he pānga rerekē i roto i te tūroro ki te momo tātaritanga rite. Na reira, me whakarite i te reira i te rata i muri i te hi'opo'a maitai, me te tino i runga i te whakaaturanga.
Varavara whakamahia māngai mō te maimoatanga o tūroro e kua i psoriasis (psoriasis) mamae i mate huka ki te pākia warowaihā waimaero ranei. Kia tūpato whakarite iwi e whai i te hītori o te mate pāwera ko reira, te tikanga o "Sotageksal". Analogues e taea ki te pehi i te tūtohutanga a te tinana ki akiaki mate pāwera hoki reira. Āta whakamahia rongoā te ki te hamani tūroro ki te kore te ngakau, e pängia ana ki depressions auau. Tūroro e kua i te infarction myocardial, whakakoi mōrea arrhythmia i roto i te fariiraa "Sotageksala".
Inenga me te maimoatanga wā
Tei runga i te pakeke o te mate ko takoto me te roanga o te therapy tarukino "Sotageksal". Tohutohu mō te whakamahi (kia whai analogs atu tohutohu mō te fariiraa) kei roto i te tūtohutanga e whai ake nei:
- horomia papa te katoa, e kore kokokiko, me ki te nui o te wai;
- Kei te whakamana Reception mō te 1-2 haora i mua i te kai;
- tango rongoā 2-3 wā i te ra.
e kore e maimoatanga wawe horopeta rā nui 80 mg (1 papa) takawhita me tachycardia. Heoi, i roto i te ngaro o te horopeta pānga haumanu hiahiatia nui haere. Āta, me te wā o 2-3 ra e whakaritea ai ki te 240-320 mg ia ra, engari anake i roto i te fare ma'i. Ko te whai hua tino ko te hua äta i roto i te inenga o te 80 mg ia wiki.
pea te horopeta mōrahi 6 papa ia tarukino ra "Sotageksal". Analogues, hoki kia kia nui haere te inenga o nei ki te whakaaro te tākuta reira tika, ka kia whakaritea takitahi. Ahakoa, ki te reira he riri ki te ora, e kore e nui ake te tapeke o te whakauru kaha 480 mg ia ra.
Ki te te manawanui reira disorders mahi mate täkihi, tīpakohia te talena maimoatanga rite te mahi o te creatinine whakawātea. Ko tōna hua (ki runga, ki te 30 mg / min), Kei te nuinga heke te horopeta ki e rua ki te wha nga wa.
hanga rua werohanga rō-uaua te ra, wehea ki e rua werohanga ampoule o 2 ml. patia i te otinga kei te āta i runga i 5-7 meneti. I roto i te maimoatanga, te mana e hiahiatia ana o te pēhanga toto, pini, o nga whatukuhu, me te pūnaha mimi, creatinine whakawātea i roto i te serum.
iteraa papû
Funds whakaritea mo te maimoatanga o enei mate:
- tachycardia, ventricular;
- Wolff - Parkinson - White;
- cardiomyopathy;
- patuki taimi halá, ventricular;
- prolapse takirere mitral;
- Paroxysmal fibrillation Atrial nga atria;
- takawhita (pēhanga toto tiketike);
- ārai me te maimoatanga o te infarction myocardial (i roto i ētahi wā).
I roto i te nui mahi waimaero tākihi, te herenga i te tākuta ki te aroturuki tonu te kukū o te taonga kaha i roto i te serum toto me ki te whakatika i te horopeta "Sotageksal" tarukino. He rite Analogs o nga tohu mō te whakauru. Ko, ahakoa tenei, ratou ake whakakapi kotahi tarukino ki ētahi atu kei te tino rāhuitia. kia puta tonu whakakorenga o maimoatanga, engari āta. Ka taea e whakatū ohorere meinga ino o te huru haumanu.
contraindications
taea e kore tonu e whakaritea tetahi kaihoko antiarrhythmic ki te manawanui, tae atu "Sotageksal". Analogs Ko te taua, e kore e taea te whakamahi e ratou i raro i nga tikanga e whai ake nei contraindications:
- hypersensitivity ranei taonga taketake idiosyncrasy he wāhanga p∂p∂ tauturu ranei;
- ngoikore koki pakohu;
- whakaiti i tohua i roto i te auau ngakau (bradycardia);
- ma'i tukanga pūkahukahu taunutia;
- nui huangō arahau;
- täkihi;
- infarction myocardial whakapeka;
- kore ngakau whakapeka ma'i ranei;
- ru cardiogenic;
- elongated QT syndrome wā ;
- tau o ngā tamariki;
- mate pāwera, Rhinitis pāwera;
- hapūtanga me te ū;
- pēhanga iti (hypotension);
- rehunga whānui;
- kikohangatia;
- mate iaia piringa;
- (Pāngia huru e atu maha i roto i nga wahine atu i roto i te tangata) te whanaketanga o te momo tachycardia "pirouette".
e kore he wheako nui ki te tarukino i roto i te hapū. Anake "Sotageksal" i whakaritea i runga i tohu faufaa. Ritenga i roto i te huatū tuatahi tū hoki he riri ki te ora fetal, a tango ratou e taea e arahi ki te materoto. raraunga rangahau pono i runga i te whakauru o te tarukino i roto i te wahine mau i te tamaiti e kore e tonu i.
I roto i nga marama whakamutunga o te therapy ka kia haeretia iti hoki 2-4 ra i mua ki te tuku, ki te te wahine e te reira i roto i te wā katoa o te hapūtanga. meatia tenei e ki te whakarite kia kore i whai i te hou te tukino o ngā mahi romahā, bradycardia ranei hypotension tika ki te tarukino "Sotageksal".
kia mutu analogues i runga i hydrochloride sotalol ki te tango, ki te he ū, he whaea taitamariki, rite te taonga e te kaha ki te tomo ki roto ki te waiu, uma me te tae nohanga tiketike reira. Ki te kia tonu tohu o te maimoatanga, he pai taua ū ki te mutu, whakakapi ranunga waiu urutau rite ki tau o te tamaiti.
pānga te taha me te tuwhena rawa
Ka taea e whai te reira i paanga kino ki te Cardiovascular, endocrine, mimi, romahā, kūnatunga me te pokapū pūnaha io whakamahi wā roa-o te tarukino "Sotageksal". meinga Analogs pānga taha rite. kia wheako te manawanui:
- hāhā o te manawa, te whakanui ake i patua angina, tohu o te kore te ngakau, mamae ngakau, vasospasm, syndrome o Raynaud ;
- whakapairuaki, ruaki, korere, puku mamae, gassing nui, flatulence, kaupapa whēkau uaua, maroke kiriuhi mucous i roto i te mangai;
- manukanuka, rōpū,, mataku whakararuraru, moemoea, waimaero nekeneke te ruruku, rongo mate, hīrere tūāhua, tremors, rohirohi, ānini, whanoke, kore o te moe ranei, hei kōrero, nui haere te momoe, moe manukanuka, korekore;
- pīkaru, keratoconjunctivitis, syndrome kanohi maroke (rawa i roto i tūroro e kakahu arotahi whakapā tonu), mumura o te taupoki io, iti iho i roto i te reka me te kakara, te mamae kanohi, photophobia, acuity ataata waimaero, rongo ranei;
- e suka (i roto i te iwi ki te mate huka);
- bronchospasm, laryngitis, tracheitis;
- urticaria, dermatitis, minamina kiri, erythema, psoriasis, angioedema, nui haere sweating;
- korekore mananga tane, te mamae i roto i ejaculation, wahine - heke libido me disorders paheketanga;
- kirika, uaua ngoikore, haehae, cyanosis o nga topito.
I roto i te take o te tuwhena rawa e taea puta:
- pehanga o ngā mahi cardiac;
- hāhā o te manawa;
- asystole, kaihapai, ngoikore, whanoke;
- cyanosis o pito;
- cramps uaua;
- bradycardia ki hopu cardiac tonu;
- ru Cardiovascular;
- bronchospasm;
- tachycardia.
Ahakoa taua tohu nui o te tuwhena rawa, he onge te mate. A, no te Me tuatahi poisoning tarukino ki te mutu tango i te rongoā "Sotageksal". Analogs me arowhānui hydrochloride sotalol tōtika putanga i te wahi gastrointestinal i muri i ingestion taero absorbent. I roto i te take o te tuwhena rawa maimoatanga symptomatic whakaaturia te. I roto i te wā o te paihana nui e tika ana lavage pekitīlia me te ruaki, mau tonu mahi ora nui o whekau. pota nui e tino nekehia atu e tātari toto. Pūkoro tukupu huka toto kia puta i roto i tūroro e piri ki te kai tino hemokai ranei.
Analogs me arowhānui "Sotageksala"
Sotalol hydrochloride roto i roto i te hua hua i roto i Switzerland ko Germany, i raro i te ingoa hokohoko "Sotageksal". Analogues E whakaaturia ona me ētahi atu taero ki hanganga rerekē, i roto i te tua ki te pānga antiarrhythmic atawhai mamae uaua, whakaiti pēhanga toto, me te whakapai ake i te mahi o te atria. Ko ētahi o ēnei:
- "Inderal" "Inderal", "obzidan", "Pranolol" (whakauru hohe - propranolol) whakamahia mo te maimoatanga o ischemia, arrhythmia me takawhita.
- "Pumpan" - kaihoko homeopathic i runga i ngā wāhanga huawhenua.
- "Magnerot" kei roto konupora orotate te whakamahia dihydrate mō te rongoā arteriosclerosis, disorders o lipid pākia.
- "Korvitol" (metoprolol tartrate) he whai hua hoki migraines.
- "Nebilet" (nebivolol hydrochloride) Kei te tohua mo te takawhita, mate rere pūroto.
- "Qudesan" (taka) - he tāpiritanga koiora e hāngai ana i runga i coenzyme Q10 mo te ārai me te maimoatanga o arrhythmias.
- "Etatsizin" (etatsizin) tono te i te tachycardia;
- "Arrhythmia" "Amiodarone" (amiodarone hydrochloride) e whakamahia i roto i te cardiac, tachycardia, arrhythmia Atrial.
- "Propanorm" (propafenone hydrochloride) whakamahia te ka ventricular me arrhythmias supraventricular.
- "Neo-Giluritmal" (praymaliya bitartrate) Kei te tohua hoki arrhythmias ventricular, tachycardia.
- "Korgard" (nadolol) te whāngai hoki i te maimoatanga o te pectoris angina, migraine.
Russia hua "Sotalol Canon" me "Tenzol" ki te taua whakauru kaha rite te "Sotageksal". Analogues i Moldova, Ukraine me whenua tata i roto i pharmacies mama atu i te tarukino taketake. Ko te utu o te raau taero tei runga i te whenua, me te kaiwhakanao. ngā rongoā kāinga te tikanga i te utu tino raro atu i ki waho.
Reviews
He ko he whakaiti nui i roto i te ärai auau i roto i fibrillation Atrial, ki te riro tonu "Sotageksal". Analogs kore e pera pai arotake manawanui. Ehara i te mea i nga wa katoa e rite taero i kamupene rerekē, ara, ki te whai ratou i te taua hanganga. He tokomaha wehi e tohu kamupene nanakia te kukū nui o whakauru kaha ia papa i te reira mau he. No te mea o tenei maimoatanga e kore e taea e kawea te hua e tūmanakohia ana. Reviews o "Sotageksale", i te rerekē, pai atu. Ia whakamahia tōtika i roto i te maimoatanga matatini o mate Cardiovascular i ngā wāhanga rerekē.
I roto i te nuinga o te wā i reira ko te whakapai ake äta i roto i te āhua whānui o te tūroro i raro ki te maimoatanga matatini. he mahuinga e rua i roto i te kapu, me te ārai i te tarukino. Whakawa i nga arotake o te tūroro ki te tātaritanga o "fibrillation paroxysmal," tauturu te rongoa ki te pupuri i manawataki ngakau noa (whakaratohia, ki te tangohia tonu te tiaki therapy). Heoi, tūroro mea kihai i e maia ki te whakaara ratou ake horopeta kahore tūtohutanga o te tākuta e tika ana ki te tūpono o ngā pānga taha nui.
e kore e pānga rawa pai i runga i te ingoa o te raau taero ētahi o te arotake. Kei te whakapono te reira e te pānuitia te reira, a e kore e taea ki te whakaora anemia, arrhythmias koiora, hypokalemia me hypomagnesemia. Kei te tuhia te reira e hydrochloride sotalol rama ke he uaua ki te kitea i roto i pharmacies rohe. Iwi tikanga ki te whakamahi i ngā wā katoa i te tikanga o ite mau fifi ki tona rironga. Na reira, i mua i te tīmata maimoatanga, kia e ka waiho reira taea ki te haere tonu hoki te wa roa.
He aha e kore e taea te ngā fariiraa "Sotageksala"
I roto i tūroro maimoatanga he reira e minaminatia ki te hoatu ake taraiwa, pahikara, motopaika. mōrearea hoki he mahi katoa e hiahia nui haere te aro me te whakamātau tinana kukū, me te arotahi. A, no te fariiraa i moni atu mō te whakaiti i te pēhanga he pea ki hypotension. Kei te riria te reira ki te whakakotahi "Sotageksal" ki taua raau taero:
- taiāki, rite kua whakanuia ana tona kukū i roto i te toto;
- katote me te raveraa ra konupūmā;
- te tikanga mo te rongoā whānui inhalation ranei;
- inhibitors Mao;
- iodine-kei roto rawa;
- Diuretics;
- pāhare ergot;
- pōuritanga tetracyclic.
E kore te te rongoā whakahaerea tukutahi ki antiarrhythmics o ahau piha me III. Kei te contraindicated ano te reira i roto i te fariiraa i taero whakapōauau, sedatives me antihistamines, antipsychotics, coumarin, relaxants. whai wāhi hoki ratou ki kaha korekore pūnaha io pokapū. arata'i rehunga tukutahi ki te pēhanga toto nui haere, me te depresses kiko myocardial. Kei te riria te reira ki te mahi i te whakamātautau kiri ki te whakatau i te momo o allergens. faarahi tenei te mōrea o te anaphylaxis, angioedema, me asphyxia.
Drug "Sotageksal" tukua i roto i pharmacies i te whakahaunga. maimoatanga motuhake o te arrhythmia e kia meinga tauhohe kino nui. Na, i mua i te tango koe i te rongoā, kia kōrero tonu koe i te tākuta.
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