HauoraMau faaineineraa

"Felodip": tohutohu mō te whakamahi, arotake. analogues tarukino

E karanga hoki te tarukino "Felodip"? Ka tohutohu hoki te whakamahi o te tarukino kia whakaahuatia i roto i te taipitopito i roto i te tuhinga aroaro. Hoki i roto i o reira, ka ako koe e pā ana ki te mea whakaritea tenei tarukino te, aha taha pānga kua reira, ahakoa ranei e kore tenei contraindications tarukino, te nui o te utu i te reira, e he analogues me pera atu.

Ko te hanganga o te raau taero, te ahua o te whakangao me te tākai

I roto i te aha puka e taea te kitea i te tarukino rongoā "Felodip"? i runga i te whakamahi o tenei aratohu rongoā kī e ko te reira e wātea ana anake i roto i te puka o papa ki te mahi auroa. Ano, pota rerekē o te tarukino he kōpaki rerekē:

  • pire kōwhai i roto i te puka o pi, kahore tetahi kakara denoted e te maha 2.5. mahi te huānga kaha taua felodipine tarukino i roto i te nui o 2.5 mg. Excipients o te tarukino he monohydrate reihuka, hypromellose, microcrystalline cellulose, waikura rino whero, povidone, Titanium hāorarua, gallate propyl, waikura rino kōwhai, stearate konupora, propylene glycol, anhydrous silica colloidal, talc. I roto i te hoko o te tarukino kaha tomo te namunamu 10 papa e kua whakanohoia i roto i ngā pouaka pepa.
  • Papa o te marama tae māwhero i roto i te āhua o pi, kahore tetahi kakara denoted e te maha 5. Ko te wāhanga kaha o taua faaineineraa protrudes felodipine i roto i te nui o 5 mg. Excipients o te tarukino protrude monohydrate reihuka, hypromellose, microcrystalline cellulose, waikura rino whero, povidone, Titanium hāorarua, gallate propyl, waikura rino kōwhai, stearate konupora, propylene glycol, anhydrous silica colloidal, talc. I roto i tomo i te hoko o te tarukino kaha te namunamu 10 papa, kua whakanohoia ki ngā pouaka pepa.
  • Papa kuratea pi parauri āhua kahore tetahi kakara whakaritea whika 10. Ko te huānga kaha o te taua mahi tarukino felodipine i roto i te nui o 10 mg. Ngaahi houalotú he monohydrate reihuka, hypromellose, microcrystalline cellulose, waikura rino whero, povidone, Titanium hāorarua, gallate propyl, waikura rino kōwhai, stearate konupora, propylene glycol, anhydrous silica colloidal, talc. I roto i te hoko o te tarukino kaha tomo te namunamu 10 papa. Opupu whakanohoia ki ngā pouaka pepa.

Ko te āhuatanga pharmacological o te tarukino

He aha te mea he pūrere hauora "Felodip"? Tohutohu mō te whakamahi o te tarukino ta e ko ia he hongere pūārai konupūmā puhoi. no raau i Tirohia ki te rōpū o te dihydropyridine.

taea ki te faaitoito pānga antianginal me antihypertensive tenei rongoā ko. I tua atu, te whakaiti reira te pēhanga (toto) na roto i te whakaiti i resistance iaia piringa.

Aha te tahi atu āhuatanga i taero "Felodip"? Tohutohu mō te whakamahi o te faaineineraa ngā pārongo e ma'u ia he pānga anti-rere pūroto horopeta-ti'aturi. whakaiti Medication rahi infarction, a hoki tiaki te tinana i fifi reperfusion.

Tenei taputapu e ngā kahore pānga kino inotropic. He he pānga iti i runga i te pūnaha whakahaerenga.

Ko te pharmacokinetics o te tarukino

Kia pehea te roa horomia te tarukino te, "Felodip"? Tohutohu mō te whakamahi, te tikanga o tenei urupare whakarato e i muri i te horopeta o medicament ki te taonga kaha te tata rawa whenumi i te wahi kūnatu me mahi tonu. Ngā mihi ki tona puka inenga, tuku roa o te huānga kaha whakarite tona kukū kākahu i roto i te toto (i roto i te ra), me hoki arata'i ki te hua i roto i te wāhanga absorption.

E kore e taea e tatou te mea e kore e te bioavailability o te tarukino whakawhirinaki i runga i te horopeta haumanu, me te he āhua 15%.

Ka herea e ki pūmua wē me te ake ïa ko reira āhua 99%. tukua te medicament te me te waiu, uma me te ô i te arai toto-roro me te arai placental. Ki te whakamahi roa o te taonga kaha puta kahore haaputuputuraa.

Hea metabolized te tarukino te "Felodip"? metabolized te whakauru kaha o tenei kaihoko i roto i te ate. I roto i tenei puka metabolites tautauā.

Ko te hawhe-ora o te tarukino ko e pā ana ki te 25 haora. teuteu whakaaturia rite metabolites (tata ki 70%) i roto i te mimi me feces (30%).

Tuhinga medicament

I roto i ētahi wā, whakaritea te manawanui te rongoā "Felodip" (5 mg) Tohutohu o tenei rongoā kei roto i te rārangi e whai ake nei o tohu mō te whakamahi:

  • takawhita;
  • angina;
  • arrhythmia;
  • mate ngakau coronary;
  • disorders circulatory;
  • syndrome o Raynaud.

contraindications taero

I roto i nei tino take riria ki te tango i rongoā "Felodip"? Reviews o tākuta, me te te tohutohu e whai kī e kore e kia whakamahia te tarukino i raro i te tikanga e whai ake nei:

  • whakapeka infarction myocardial, me te i roto i te marama kotahi i muri i myocardial;
  • angina iu;
  • ru cardiogenic;
  • kore ngakau, rawa decompensated;
  • stenosis te pūtahi o (hauora nui);
  • hapūtanga;
  • hypotension (nui);
  • i roto i ngā tamariki me ngā taiohi (i raro i te 18 tau);
  • i roto i te hohipera;
  • nui haere te tūtohutanga o te manawanui ki te tarukino atu pārōnaki dihydropyridine ranei.

e kore e wareware tetahi e tenei taputapu ki te tūpato tino whakaritea ki tūroro ki iti hoki ate, me te tākihi.

pūrere Medical "Felodip": tohutohu mō te whakamahi

Ka kia te aroaro he iti atu analogues o tenei taputapu. Na e hiahia ana ahau ki te korero ki a koutou e pā ana ki te āhua o te rongoā kia tangohia tika.

A, no te takawhita whakaturia horopeta mō ngā pakeke me te iwi paari te takitahi. Tikanga, te nui tuatahi o te tarukino ko 5 mg kotahi te ra. I roto i te kōwhiringa o ngā tūroro e tika ana tūtohutia te inenga e ki te whakamahi i te papa o 2.5 mg. A, no te Me te akiaki ki te whakapiki ake i taea te horopeta o rongoā kia. Ko te rōrahi toharite o te medicament mo te maimoatanga tiaki o 5-10 mg ia ra.

Hoki tūroro paari tūroro ki te mahi ate waimaero i roto i te therapy tarukino wawe ranei whakahaerea nei i roto i te nui o 2.5 mg ia ra.

I roto i te rongoā angina eu "Felodip" whakaritea takitahi. Ko te kupu tona horopeta tuatahi (mō ngā pakeke), ko te 5 mg kotahi te ra. Ki te hiahiatia, e taea te nui haere te horopeta ki te 10 mg ia ra. Ko te nui mōrahi rā o te tarukino ko 20 mg.

Papa "Felodip" tukua te ki te tango i roto i ngā ki inhibitors ACE, beta-blockers me Diuretics. Heoi, kia tuhia te reira e ia whakarei te pānga hypotensive te. Na reira kia koe tino tupato no o te nui haere tūpono o hypotension.

I roto i te tūroro ki te mahi ate tino waimaero kia heke te horopeta o rongoā.

Tuku e te tarukino kia anake e tangohia i roto i te ata i mua i te parakuihi. I roto i tenei take, ki te papa i roto i tetahi take e kore e taea anganga, kuru wehenga ranei.

tikanga tuwhena rawa

whakamahi hē o pire "Felodip" kia puta te tohu e whai ake nei o te tuwhena rawa i roto i tūroro: bradycardia me hypotension (nui).

I roto i te take o te takanga o taua tohu therapy symptomatic. Ki te homai e hypotension (nui) tūroro i te tūnga whakapae, me te ara waewae. Ki te whakaute ki bradycardia, i nei take i te atropine manawanui intramuscularly whakahaere i te inenga o 0.5-1 mg. Ki te tika, ki te whakapiki ake i kawea te rōrahi o te wē e whaowhia te i ki te konutai pūhaumāota, otinga kūhuka dextran ranei.

A, no te whakaritea nga mehua koretake i runga-whakaahuatia rongoā ki te manawanui ki te pānga matua i runga i receptors alpha-adrenergic.

pānga te taha i te tango i te raau taero

E ahei ranei i te pānga kino i runga i te tinana tangata tango i te rongoā "Felodip"? Analogues o tenei taputapu me te faaineineraa iho maha ai ānini, Makere kanohi, whanoke, palpitations me te rohirohi. Heoi, kia tuhia te reira e e reversible taua tauhohe. Ratou te tikanga puta i te timatanga o te therapy, me te e whakanui ake i te inenga o te tarukino.

E te ara, i runga i te nui kei riro rongoā kia puta te manawanui me te edema piringa. E ai ki te tohunga, he ratou te hua o te vasodilation precapillary.

I roto i te tūroro ki te periodontal mate kapia ranei i roto i ngā tūroro i te fariiraa i te tarukino pea he puku iti o te pae. Ka taea te te ārai i tēnei tukanga, ki te puritia e koe te akuaku waha tino.

I roto i ētahi wā e whakaaro tatou fariiraa i rongoā riro te take o te pānga taha e whai ake nei:

  • pūnaha Cardiovascular: palpitations, tachycardia, me edema piringa.
  • tauhohe Dermatological: photosensitivity, pruritus, urticaria.
  • pūnaha io piringa, me te puku o: paresthesia, ānini me te whanoke.
  • pūnaha musculoskeletal: arthralgia, myalgia.
  • wahi kūnatu: hyperplasia gingival, whakapairuaki, hua i roto i whākōkī ate.
  • Ētahi atu: rohirohi, tauhohe hypersensitivity, tae atu angioedema.

Analogs, me te utu o te tarukino

Kia pehea te nui Ko te rongoā i mua i a tatou? Ko i te whakahaerea te take i whakaarahia e te maha tūroro pangia tenei maimoatanga. Me kï reira e taea te hokona he rongoā i te utu e whai ake nei i teie mahana, ko te:

  • Papa o 2.5 mg (30 nga wahi) - 425 moni Russian;
  • papa i roto i te rōrahi o te 5 mg (30 nga wahi) - 556 moni Russian;
  • pire i roto i te rōrahi o te 10 mg (30 nga wahi) - 831 moni Russian.

He aha e taea e whakakapi i te tarukino "Felodip"? E wātea ana Analogs o tenei tarukino i roto i tata rongoā katoa. I roto ia ratou, e hiahia ana ahau ki te whakanui i nga rongoa e whai ake nei: "Plendil," "Felodipine-NW", "Felodipine" me "Felotenz ia faataere".

urupare pai i tūroro e pā ana ki te hua rongoa

Mua e pā ana ki "Felodip" āhua faaineineraa e ko reira tino whai hua, me te pai noatia-e tūroro, ahakoa o tau me te ira tangata. I tua atu, kia tarukino kaha kia tangohia noa e tūroro ki te mate huka, disorders tākihi, huangō me te tahi atu mate pūkahukahu taunutia ki syndrome o Raynaud, hyperlipidemia, kauti, me i muri i tana pukapuka transplantation.

tohu maha tohunga i te meka e te rongoā e kore pānga i runga i te kōtaha lipid me kūhuka i te toto kukū.

arotake kino

I roto i te arotake kino e waiho tūroro i runga i tenei tarukino, ka taea e tatou mōhio te hunga e pā ana ki te utu nui o te tarukino. Ahakoa tautohe taka rongoā e he tino hāngai ki te pai, me te kounga tona utu.

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