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"Flyuanksol": tohutohu mō te whakamahi, tākuta tūturu. pānga taha "Flyuanksola" analogues o te tarukino

He aha te mea te tarukino "Flyuanksol"? E whakaahuatia tohutohu mō te whakamahi o te raau taero, ona kai, ngā pānga taha, te puka tuku, me ngā āhuatanga pharmacological i roto i taipitopito i roto i tenei tuhinga. Mai i reira ka ako koe e pā ana ki te mea ka mea nga contraindications me tohu kua te raau taero, te nui o te utu i te reira, te mea e tupu i roto i te take o te tuwhena rawa, a na i runga i. D.

Ko te hanganga o te tarukino me ona puka tuku

He aha te mea te taonga kaha kei te rongoā "Flyuanksol"? kī tohutohu mō te whakamahi o te ako medicament e rite wae kaha protrudes reira hydrochloride flupenthixol.

Ka rite ki ki te ahua o te tuku, engari i tenei ra ko te reira e taea te tikanga e kitea anake i roto i pata, papa me te otinga, he hāngai te hinu-, tikanga hoki whakahaere intramuscular. hokohoko te tarukino tuatahi i roto i te karaihe zatemennom 10 ml, he tuarua - i roto i te kātene 100 ranei 50 me te tuatoru - i roto i ampoules o 10 nga wahi.

āhuatanga General o te tarukino

He aha he rongoā "Flyuanksol"? E te aroaro Mua e pā ana ki tenei tarukino i raro. Papa me te werohanga ko te rōpū o antipsychotics. riro ratou anxiolytic, raau, me te pānga whakarokiroki. Pai urupare e pā ana ki tenei tarukino i roto i ngā mōhiohio e tōtika ai whakahohetia te āhua aronganui o te manawanui, me te whai wāhi ki te urutaunga pāpori.

Ko te āhuatanga pharmacological o te tarukino

He aha e nga āhuatanga o te tarukino pharmacological "Flyuanksol"? Tohutohu mō te whakamahi kōrero e tenei tarukino ko te neuroleptic, ārai receptors adrenergic me receptors dopamine i roto i te roro. Ka rite ki te hua o te taonga kaha tutuki te whakarokiroki. Tikanga, puta tenei i runga i te inenga auau 8-ra.

He aha e tūroro e pā ana ki ngā rongoā "Flyuanksol"? Reviews o tūroro i roto i te rota o ngā mōhiohio. I roto i te nuinga o te wā, mōhio ratou e te raau kaua hohoro faaore tohu o āhotea, ngā paheketanga, me te whai wāhi ki te faaho'iraa mai o te whakaaro. Tūroro nei nga disorders ngaahi fasí ', he whakahoahoa me te urutau ki te hapori.

āhuatanga rongoā

Nahea te tarukino "Flyuanksol"? Reviews o tākuta me ētahi atu ngaio mea e te āhuatanga o tenei tarukino ko e, i runga i te horopeta kei taea mahi i te reira i runga i te manawanui i roto i ngā huarahi rerekē.

faaite pānga ähotea i muri i te tikanga tono medicament i roto i te nui o 3 mg ia ra. E te ara, e faarahi te kaha o te pānga ki te inenga.

Ko te nui ki te 25 mg ia tarukino ra kahore pānga whakarokiroki. Heoi, kia tuhia te reira e i pota teitei, e taea ai te pānga whakarokiroki kore-motuhake.

I roto i te awhe horopeta tohua kaihoko neuroleptic he pānga anxiolytic korerotia. A, no te whakamahi i pota iti (ki runga, ki e pā ana ki 3 mg ia ra), kia mahi i te tarukino rite te rongoā raau tikanga.

Ko te kupu, taea ki te whakaiti i nga tohu matua o te āhotea, tae atu ki ngā whakaaro horihori Wairau, moemoea me whakaaro whakararuraru, te tarukino "Flyuanksol" ko. He āhuatanga disinhibitory (i.e. whakahohe me antiautisticheskim) me te whakaiti i te mate te tūāhua, e te mutunga whakatairanga faaitoitoraa o tūroro ki tohu fakalotofo'í, whakahaere ratou urutaunga pāpori, me te whakarei ake sociability.

Ētahi atu e pā ana ki te puka injectable

Te faaineineraa "Flyuanksol Depot" Ko te otinga hinu tikanga hoki werohanga taupuni intramuscular. I roto i te mau parau te tahi atu, whakatakotoria tenei raau te puka flupenthixol.

A, no te whakamahi i tenei otinga i roto i pota iti, me te reo (ki runga, ki te 100 mg katoa ra 14) ki te manawanui e kore he whakarokiroki unspecific. Ahakoa reira Kei te tipu haere tonu i pota teitei.

He aha tohunga te mea e pā ana ki tenei ahua o te tarukino ( "Flyuanksol Depot")? Reviews whakarato e te otinga taua he roanga roa o te rongo ki te manawanui, kaua ki te papa rongoā. Ano, whakawhetai ki a ia, he mea ohie ki te kawe i roto i te maimoatanga ähotea tonu, i te mea tino nui mō ngā tūroro e kore e kawe i roto i whakahaunga hauora.

Mai i te runga ake e taea te faaoti i te reira e taea ana ki te ārai i relapses auau e pā ana ki arumanga māhorahora o therapy te tarukino "Flyuanksol Depot" ko. werohanga Intramuscular taea te kawea atu i wā o rua ranei wha wiki.

Pharmacokinetics

pire Kia pehea te roa kua horomia "Flyuanksol"? I muri i whakahaere waha tutuki te kukū mōrahi o te pūmotu kaha i roto i pā ana ki 3-7 haora i roto i te wē. Ko te bioavailability o te tarukino ko 40%.

huānga tarukino Active paku te ô i te arai placental. Me mahara hoki käore te reira e, i roto i te moni iti, te miramira reira ki te waiu o tona whaea. Ratau, te metabolites i mahi neuroleptic.

Nahea werohanga "Flyuanksol Depot"? kī Guide e muri werohia intramuscular o taonga cis (Z) te whakamamaetia decanoate -flupentixol wāhinga (enzymatic). ngā tenei te āhuatanga kaha o te cis (Z) -flupentixol me te waikawa decanoic. tutuki te kukū mōrahi i roto i te serum te tuatahi i te mutunga o te wiki tuatahi i muri i werohia.

A, no te fariiraa i te papa ki to ratou wā tupuranga ko e pā ana ki 35 haora. Ki te reira i whakamahia he otinga mo te werohia, heke ē te kukū i roto i te serum (i muri i te 3 wiki).

Whakaaturia medicament kaha i roto i te puka o metabolites roto i te whēkau, me whatukuhu.

Tuhinga mo te whakamahi o āpiha neuroleptic

I roto i ētahi wā, whakaatu ana te tarukino "Flyuanksol"? kia rerekē tona mahi, i runga i te inenga rānei.

tohua te tarukino te i pota ake ki 3 mg ia ra mo te tikanga pathological e whai ake nei:

  • whārua ngawari me te tohu āhua, haere tahi i te ngenge, te manukanuka, me te kore o te kaupapa;
  • disorders psychosomatic e faaite mai ki tauhohe asthenic;
  • disorders pōhewahewa (tonu), haere tahi i te tau'a, whārua me te manukanuka;
  • a koi disorders manukanuka-a, me te te āhua o te ahotea aronganui nui, e kore e rapua e te whakarokiroki pānga hypnotic ranei (hei tauira, ki te te te manawanui memeha tranquilizers).

Medicament "Flyuanksol", analogues o nei e kia te aroaro i te mutunga o te tuhinga kua whakaritea, i toketaá o 3 mg ia ra me te ake ki te reira ko te ine o te whai ake: tikanga psychotic e kua haere tahi e horihori Wairau, moemoea, raruraru i roto i te whakaaro, anergy, tau'a me te autism.

Contraindications ki te whakamahi o āpiha neuroleptic

I roto i ētahi wā, e kore e tūtohu ana ki te whakamahi i te tarukino "Flyuanksol"? Tohutohu mō te whakamahi ngā te rārangi e whai ake nei o contraindications:

  • tau o ngā tamariki (18 tau);
  • CNS korekore;
  • hohipera;
  • i roto i te hapū;
  • haurangi (koi) barbiturates;
  • hinga;
  • haurangi Pë opioid whakapeka;
  • pheochromocytoma;
  • poisoning whakapeka waipiro;
  • āhua comatose;
  • wheua whakaīngoatia wheua;
  • huringa pathological i roto i te toto;
  • hypersensitivity ki neuroleptics he hanganga tioksantenoviy.

Me mahara hoki käore te reira e kore he mea tika ki te whakahau i te tarukino i roto i pota iti (ki 3 mg) i roto i te āhua o te te totoa excitations ranei.

Drug "Flyuanksol": ako (papa, makaka)

Hoki te maimoatanga o te manukanuka, me te fakalotofo'í disorders kia te horopeta tuatahi o te medicament i roto i te papa 1 mg kotahi te ra (he pai i roto i te ata), ranei 500 mcg rua rā. Ki te he ngaro te pānga haumanu, ka taea te nui haere te nui o te tarukino i roto i te wiki ki te 2 mg. Ko te kupu kia wehea te inenga rā (2-3 mg) ki te maha o ngā wāhanga. Ki te he ngaro te pānga, ka whakamahi i te raau taero i roto i te horopeta maximal (i.e., 3 mg), ka kia kia memeha reira.

I roto i te maimoatanga o ngā āhuatanga psychotic whakaturia nui o rongoā takitahi anake. kia te inenga o ia rā tuatahi 3-15 mg i roto i te 3 werohanga wehea. Ki te hiahiatia, e taea te nui haere te rōrahi mea ki 20 30 ranei mg ia ra. E kore e te inenga mōrahi e neke atu i te 40 mg.

Ka rite ki whakahaerea fakafofonga'i kaihoko tiaki maimoatanga e i roto i te nui o 5-20 mg kotahi te ra (i roto i te ata).

Ko te maturuturunga iho "Flyuanksol", kia anake ratou kia tangohia roto. Doctors te nuinga whakahau te tarukino i roto i tenei puka anake i roto i te take ki te, no te mea katoa te take, e kore e taea te tango i te rongoā waha (papa). inenga tautoko mō ngā tūroro he 4-40 mg ia ra.

Werohanga "Flyuanksol": ako, arotake manawanui

Me whakahaere te otinga hinuhinu mō werohanga taupuni intramuscular hohonu ki te hautahi waho o runga o te papa. kia anake kia tāuta inenga me te wā i waenganui i maimoatanga takitahi (motuhake o te pānga haumanu).

Kei te nuinga o tenei waihanga whakamahia i roto i te nui o 20-40 mg (ranei 1-2 ml) katoa 2 ranei 4 wiki. Me kï reira e kia rapua e te tahi mau tūroro pota nui me te wā poto i waenga i werohanga.

Ki te te rōrahi whakaritea o rongoā mō te werohanga (20 mg / ml) he neke atu i te 2 ranei 3 ml mo te 1 tukanga, he mea e tika ana ki te haere i runga i ki te otinga o te kukū tiketike.

Te faaineineraa o te 100 mg / kia ml kia patia i roto i te rōrahi o 50-200 mg (ranei 0.5-2 ml) katoa 2-4 wiki. I roto i te matahoki whakapeka ranei exacerbation o te mate ētahi wā titau te tikanga he whakataki kotahi-wā i roto i te nui ki runga ki te 400 mg i wā o 2 ranei 1 wiki. I muri haere nga tohu whakapeka, me hua e koe he whakaiti āta i roto i te inenga ki te tiaki (20-200 mg katoa 2-4 wiki).

Ki te hiahiatia ki te haere i te ahua-waha o te tarukino hoki parenteral faaineineraa therapy tautoko, e tūtohu ana ki te kia i runga i te kaupapa e whai ake nei:

  • nui ia (i roto i te mg) o te tarukino i roto i te papa x 4 = inenga kotahi (i roto i te mg) werohia nga ra 14.

Me mahara hoki käore te reira e roto i tetahi wiki i muri i e tohutohu whakahaere o te tarukino ki tango i te raau taero i roto i papa tonu, engari i te horopeta raro. A pee i-ake rōrahi me te āputa i waenganui i te ngā tukanga whakapumautia i roto i runga i te pānga haumanu.

inenga mōrahi otinga injectable (kotahi-atamira) Ko e pā ana ki 400 mg. Ko te kupu kia te āputa i waenganui i werohanga i te wiki.

E ai ki ngā whakautu o te tūroro, ka whakamahia tika, te faaineineraa, me te haapa'oraa o tūtohutanga hauora, te mea he pānga pai i runga i to ratou ahua aronganui whānui.

pānga taha

E ahei ranei i te pānga kino i runga i te rongoa tinana "Flyuanksol"? e kitea ngā pānga taha i roto i te raau taero, ahakoa o tona ahua. Tenei e ratou i teie nei.

  1. pūnaha Nervous: giperkinetiko-hypertensive syndrome (marama extrapyramidal), ngoikore, akathisia, rohirohi, whanoke, whakamātau tinana retardation, dyskinesia tardive, tauhohe takawiri me neuroleptic syndrome mārere.
  2. Ngakau me te toto oko: tachycardia, hypotension, orthostatic.
  3. pūnaha hematopoietic: granulocytopenia.
  4. whēkau Sense: ngangau o noho.
  5. GI: kōroke, jaundice cholestatic, mangai maroke, huringa rangitahi i roto i ngā whakamātautau mahi ate.
  6. pūnaha endocrine: taonga taimaha, galactorrhea, sweating, gynaecomastia, paruparu, dysmenorrhea, nui haere te hiahia, heke libido, hiko wera.
  7. pūnaha mimi: pupuri mimi.
  8. Mate pāwera: dermatitis, photosensitivity, me ponana kiri.

tohutohu motuhake mō te whakamahi

Ki te rongoā tūpato tino whakaritea ki tūroro ki disorders Cardiovascular, disorders takiri, kore romahā, papahewa, mate a Parkinson, mariao puku me paru 12-tiperstnoj, huangō, waipiro, emphysema, te pupuri mimi, kore ate, me te benign prostatic hyperplasia.

Ki te mea kua riro i mua i te manawanui neuroleptics tranquillizers ranei ki pānga whakarokiroki, he mea e tika ana ki te mutu tango ratou pai.

A, no te maimoatanga wā roa-, rawa i toketaá tiketike mana tūtohutia me arotake huru o te manawanui i roto i te tikanga ki te whakatika i tiaki horopeta.

I roto i te maimoatanga tukutahi o taumahi huka o mea kia rapua e waihanga nui te ako o te taiāki.

I roto i te tono o neuroleptics kia whakawhanake syndrome mārere neuroleptic. Ko tōna tohu matua he uaua rigidity, tūāhuruiti, rereke te mana hinengaro, me te pōrearea o te pūnaha io autonomic. A, no te rapu taua tohu whakakorenga akiaki o te whakarite o te tarukino me te tautoko maimoatanga symptomatic.

I roto i te nuinga o te wā, rongoā "Flyuanksol" e kore e meinga whakarokiroki. Ko, ahakoa tenei, he mea e tika ana ki te tango i ki pūkete ona pānga pea i runga i te kaha ki te whakahaere humarie te mīhini, ētahi atu pūhanga ranei. hiahia ana ano ahau ki te mōhio e i roto i therapy (rawa i roto i te timatanga), tūroro kia karo mahi pea mōrearea (ki te whakatau i te whakautu ki te tarukino).

take o te tuwhena rawa

Ki te tangohia te rongoā te tika (nui haere rōrahi), kia puta ai tuwhena rawa. I roto i tenei take, whakaaturia te āhuatanga e whai ake nei: hypo- tūāhuruiti, te momoe, haehae, ranei mate extrapyramidal, ru, hypotension me te pōroa.

Aha ki te mahi i roto i te āhuatanga i taua? Ko reira e tika ana ki te kawe i roto i te therapy tautoko, me te symptomatic. Ki te i ingested te raau taero, te hiahia ki te hohoro horoi i te puku, me te ki te tango i te sorbent. I tua atu, he mea tino nui ki te tautoko i nga mahi o nga oko, te ngakau me te pūnaha romahā. E kore e tūtohu ana ki te whakamahi i epinephrine rite kia arahi ai ki te pēhanga toto whakaiti. Ko taea tohu Extrapyramidal ki te aukati i te tarukino "Biperiden" me haurangi - "Diazepam".

Ngā pāhekoheko ki ētahi atu taero

A, no te whakamahi i tetahi-wā o medicament mea kia rahi roa'tu, ai pānga whakarokiroki o barbiturates, te waihā, me ētahi atu āpiha e whai pānga inhibitory i runga i te CNS.

Te faaineineraa "Flyuanksol" e kore e tūtohu ana ki te whakamahi i roto i te taha ki te guanethidine me Drug taonga ki te pānga rite. Tenei meka Ko e tika ana ki te meka e kia tino ngoikore ai antipsychotics ratou pānga antihypertensive.

Ki te kotahi-whakamahi medicament "Flyuanksol" Ka taea e whakaiti i te reira miramira o te tarukino "levodopa" me ētahi atu āpiha adrenergic.

I te wa ano tango i te tarukino ki te "piperazine" me "MCP" tino whakanuia ana te mōrea o te whakararuraru, extrapyramidal.

Me mahara hoki käore te reira e kore te tikanga kia konatunatua te tarukino neuroleptic aroaro rite te otinga mō te werohanga i roto i tetahi take ki ētahi atu fluids.

Utu me analogues o te tarukino

Kia pehea te nui Ko te tarukino "Flyuanksol"? Ko te tino nui tona utu. Na, mo te 50 papa o te 1 mg o koutou e whai ki te utu e pā ana ki 500 moni Russian. Ki te hiahia koe 100 papa 5 mg, e taea te hokona ratou mo 1,200 moni. Ko te ahua injectable o te tarukino, he reira noa atu te utu. Neke atu i te 10 oko (20 mg / ml) taka rongoā rapu e pā ana ki 2300 moni.

He aha te ki te taea ki te hoko rongoa "Flyuanksol" te manawanui ko te? Ko tōna analogues e hokona i roto i tata katoa mekameka rongoā. I roto ia ratou Ko te whai ake:

  1. Ko te otinga "Flyuanksol Depot". Ko reira tere me te ake kaha tarukino. Heoi, ko reira papa nui atu te utu.
  2. "Klopiksol" rongoā. I roto i te uara he tata rawa ki te taketake. haere te reira i runga i te hoko i roto i te papa, me te kua he torutoru contraindications.
  3. tikanga "Truksal". Hokona i roto i te papa. Ko te painga matua i roto i te manakohia o tona whakamahi mō ngā tamariki ki te 3-tau. Utu paku i runga i te taketake.

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