HauoraMau faaineineraa

"Olanzapine": analogues, whakaahuatanga tarukino, tohutohu hoki te whakamahi

Hoki te maimoatanga o te wairua tuakoi me te mate pourua whakamahi taero i runga i te pūtake o te taonga olanzapine. He maha taero ki ngā ingoa hokohoko rerekē, engari te pānga ähotea taua. Ko tētahi taua tarukino ko roto i tarukino "olanzapine" analogs i roto i tona hanganga te katoa whakauru hohe.

Whakaahuatanga o te faaineineraa

mahi tenei e te kaihoko ähotea "ALSI Pharma" ZAO rite te papa kōwhai marama, te āhua o e rite te biconvex rango. He he he rongoa i roto i wha toketaá. Papa ia horopeta rerekē whakairo waho tuhituhinga. Hoki inenga o 0,0025 go o te tuhituhinga whakaratohia «L», ki horopeta 0,005 go o te ti'araa «FA20». E whaowhao Papa ki 0,0075 go o olanzapine «F20C», engari ki 0.01 go o whakauru kaha Kei «N30C».

Ko te hanganga o te tarukino hanga kai hohekore, e ngā momo microcrystalline cellulose, monohydrate reihuka, filler krospovidonovy, stearate konupora. faarahi ratou tokomaha i roto i rua, e toru ranei, e wha nga wa, i runga i te olanzapinovoy inenga rānei.

Kua Kikī nga papa pota katoa o 7 mongamonga i roto i te opupu i roto i te mōkihi e taea e 4 8 ranei nga wahi.

pā ana te tikanga o "olanzapine" Taupānga Kaiwhakamahi ki te taero neuroleptic ähotea e whakaatu hunaonga mo te serotonin, dopamine, muscarinic, adrenergic me histamine hanganga receptor.

Tīpakongia iti mahi excitatory o nga neurons dopaminergic mesolimbic, he iti mahi i roto i te pūkawe karere striatal, e regulates te mahi o te pūkaha. Te heke haere te kaha i roto i te reflexes tiaki tikanga, ki te whakamahi koe i te inenga iti kahore ai moe cataleptic.

Medicine "Olanzapine" faarahi te miramira anxiolytic o te mahi whakamātautau "anxiolytic" i i rere i te reira. E waha ana tohu withdrawal, me te hua kino rite horihori me i kitea hallucinatory.

Aha whakamahia te

Papa "olanzapine" pānga puta i runga i te kāwanatanga wairua tuakoi te i roto i te pakeketanga i roto i te wähanga whakapeka, rite te pupuri me te maimoatanga protivopovtornogo roa. E whakamahia ratou hoki te whakararuraru, psychotic ki te tohu hua o horihori, i kitea hallucinatory me tohu kino pērā i flattening aronganui, te whakaiti i te mahi hapori nui, kēkeno o te taputapu waiata.

to'o Drug hohokitanga o hukihuki ki te whakararuraru, pourua, ki te pai hamani te papa wāhanga härukiruki.

Te faaineineraa "olanzapine" tukuna ngā pakeke ki disorders pourua i te puka o te monotherapy ranei i roto i te taha ki te medicaments kei roto katote lithium waikawa valproic ranei. whakamahia te tarukino te ki hamani whakapeka puka härukiruki whakauru ranei o mahi e kia puta āhuatanga psychotic, me te whai i te wāhanga huringa nohopuku.

Tikanga ngā ki ngā rongoā fluoxetine mō ngā āhuatanga fakalotofo'í e kua pā ana ki te whakararuraru, pourua.

Ngā ritenga whakamahi

Medicine tono "olanzapine" Kaiwhakamahi taunaki ana te ra i 0,005 ki te 0.02 g waha kahore pipiki aratau mana.

āhua wairua tuakoi tūroro pakeke tukinotia ki te inenga tuatahi rā o 0,010 g

nekehia mania whakapeka Pakeke, whakararuraru pourua āhuatanga e, nui rā o te olanzapine i 0.015 g, e whakahaerea nei kotahi. Ki te papa whakamahia mō te pānga pupuri te taha ki te rongoā e hāngai ana i runga i lithium katote ranei waikawa valproic, ka whakahaere i roto i te inenga rā o 0,010 g ia kotahi.

tukanga fakalotofo'í i roto i te pakeke mate pourua tika, atawhai nui ia o 0,005 g, kua ngā ki 0,020 g fluoksetinovogo taonga. Ki te kahore he he hiahia, ka tukua whakatikatikanga o dosing o ngā rongoā.

Hoki tūroro kaumātua ki taea riri nui iti hoki tākihi ki te ate ma'i ranei rite ina i reira he tūponotanga e pā ana ki te ira tangata wahine, taipāpā tau-ka heke utu whakapōturinga olanzapine tona nui rā tuatahi te ki 0,005 g

enei taputapu

Medicament "Olanzapine" ritenga he ingoa hokohoko rerekē. E whakaputaina ratou e rua kaihanga kāinga me te ke.

I roto i te kamupene Russian o taero Technologies kamupene whatu-atu ' "ki te tarukino" Olanzapine-TL ", i roto i te puka papa pani 0,0025 g kiriata.

Ētahi atu rongoā kāinga ko te tikanga o "Olanzapine", hangaia e JSC "Te Tai Tokerau Star". He he he papa ki te paninga kiriata me te horopeta o 0,005 g

wheketere Russian hua "Kanonfarma Production" JSC te tarukino "Tumau o olanzapine."

rongoā Iseraela he rongoā "Olanzapine Teva," kamupene hanga "Teva rongoā Enterprise Co., Ltd.".

orotahi Slovenian Ko te tikanga "Zalasta Cu ripa", i roto i te papa o 0,015 g mo te resorption. Hanga e te hinonga "Krka, Novo mesto." Hoki raraunga whakaputaina e te tarukino papa "Zalasta".

whakaaro orotahi tarukino Swiss te "Zyprexa" rite te lyophilisate i nga oko, i nei te otinga rite mo te whakahaere intramuscular, he horopeta o 0,010 i roto i te puka papa dispersible 0.005 karamu vai tarukino "Zyprexa Zidis". E hua ratou i "Eri Lilly Vostok SA". I roto i te mākete ho'oraa reira he "Zyprexa Arere" haapae atoa paura medicament 0,21 g

kamupene Polish o "Polpharma" rongoā hangaia "Normiton" papa ki te paninga takotoranga o 0.005 g

Drug "Olanzapine" ritenga Hungarian whakaputaina e "Kiriona Richter" i huaina papa "Parnasan" me rongoā tipu "EGIS" whakawhanakehia tarukino "Egolanza".

Whakaahuatanga "Zalasta" tarukino

E pā ana tēnei ki te neuroleptic ähotea. papa kōwhai Light e tawhio, āhua paku biconvex ki pāti pouri. E ono toketaá: 0,0025 g, 0,005 g, 0.01 g, 0,015 g, me te 0.02 go o olanzapine. wāhanga atu whakaaro Cellactose paruparu, māngaro pregelatinized me witi puka, dehydrated aerosilovy whakauru, konupora stearate.

Hei tohu i te puka papa whakaahua ana "Zalasta" ā-ako te momotuhi i roto i te puka o tuhi ki te tohu o te inenga. pōkai Kiritaki He pereti contoured 7 papa. kia roto i te mōkihi 4 8 o taua opupu ranei.

Tenei māngai neuroleptic whakaaturia ngā mahi pharmacological whanui. pānga ähotea e pā ana ki te momo ngā interlock dopamine receptor. mahi whakarokiroki meinga e te pae adrenoceptor braking e riro te hanganga reticular i te pūtau o te kakau roro.

Ko taea mahi Antiemetic i mutu D 2 receptor -dopaminovogo wahi i roto i te rohe keu-momo kei nei i roto i te pokapū hiaruaki.

kawea tūranga Hypothermic te roto e ārai i te ngā dopamine receptor o te momo i roto i te hypothalamus.

fokotuu Medicine "Zalasta" ā-ako whakamahi i faaiteraa wairua tuakoi. E taea e ki te pupuri i kaha nga huringa o ngā tohu haumanu i roto i te maimoatanga o te tūroro ki te pānga pai tuatahi i runga i te tarukino wā roa-papa.

Tikanga whakakore mania wā i roto i te puka waenganui matatini ranei. Papa whakahaere whakatupato whawhe tāruarua pokenga ki te whakararuraru, pourua i roto i te iwi ki te wāhanga härukiruki.

tikanga te tarukino te mo te whakahaere-waha kotahi te ra. e kore e matūriki kai pā te tukanga absorption o olanzapine, e taea ai e koe te whakamahi i te papa i tetahi wa. Ki runga ki whakakorenga o te tarukino āta kia whakaiti i te horopeta.

Hoki te maimoatanga o disorders wairua tuakoi te whakamahia i roto i te dosing tuatahi o 0,010 karamu ia ra.

Wāhanga o te mania timata tukinotia horopeta ia rā o 0.015 g, i whakahaerea nei i roto i te kotahi tono 0,010 karamu ranei ka ngā ki ētahi atu neuroleptics.

kawea ārai tāruarua o te whakararuraru, pourua i roto i te taahiraa attenuation i roto i roto i te hono tokonaki medicament tuatahi 0,010 karamu ia ra. Ki te tango te tangata i te taputapu i roto i te whakatutuki mania wā, mo te pupuri o te therapy te whakamahi i te taua horopeta. He mea tika ki te whakapiki ake i te nui o tarukino i te hui o te mau faaiteraa fakalotofo'í wā hou whakarōpūtia ranei, me te ki te tāpiri i te maimoatanga o te faahuehueraa huru.

Ko te horopeta rā o medicament ki te whakakore disorders wairua tuakoi, wāhanga härukiruki me disorders pourua whakatupato tāruaruatanga whakamahi i 0,005 ki te 0,020 g, te uara o e tei runga i te tawhā haumanu o te manawanui.

Kei te kore tohutohu, Heoi, ka kia tono ruhiruhia raro inenga tuatahi o runga ki te 0.005 g taua mahi ki tūroro i te 65 tau o te tau, ki te reira he āhuatanga mōrearea.

Whakaahuatanga "Olanzapine Canon" tarukino

mahi ähotea Active o rongoā neuroleptic e wātea ana i roto i te puka papa pani ki te takotoranga. Ko te āhua o te papa häunga ki e rua papa ohu kōwhai, te tirotiro ā-o te tae kotahi.

vai te reira i roto i rua toketaá: i 0,005 g, me te 0.01 go o olanzapine. Ko te kai ngaahi houalotú ngā cellulose hydroxypropyl ki whakauru iti, konupūmā hauwai Phosphate, te konutai croscarmellose, mannitol, konupora stearate.

i hanga takotoranga kōwhai kiriata Opadry te o te momo tuarua, polyvinyl waipiro, macrogol, talc, Titanium hāorarua, rino waikura.

maimoatanga Drug whakaritea mo hauā, mō te pupuri me te tono antirelapse roa tūroro pakeke e mate ana i disorders wairua tuakoi.

kawea te rongoa te monotherapy me huinga tīaroaro ki te pūhui konukōhatu ki te ahua kaha o te wāhanga härukiruki whakauru ranei o te mate aronganui pourua, e he kīanga ki ngā wāhanga nohopuku huri psychotic me ki. Medicines ki te ārai i aua i roto i te iwi ki te disorders pourua, ki te i āwhina te tarukino ki akakoromaki i te atamira härukiruki.

I roto i te maimoatanga o ngā pakeke ki te korekore meinga e te whakararuraru, pourua, me te pūmau rongoa tohu fakalotofo'í "Canon Olanzapine", he neuroleptic, kia ngā ki māngai kei roto fluoxetine.

Kei te mau te reira i-waha, e kore piri ki te kai. E taunaki ana Guide e te inenga haumanu o te medicament, i te mea he ra, kua tīpakohia takitahi te maha o 0,005-0,020 tikanga mo ia manawanui i runga i nga tohu haumanu rānei.

disorders wairua tuakoi manawanui pakeke hamani tuatahi rongoā dosing ia i roto i 0.010 g, e whakahaerea nei i kotahi.
Herenga te whakararuraru, pourua mania whakapeka faaore i te inenga o ia rā o te tarukino ki 0,015 g 0,010 go o olanzapine ngā ki āpiha kei roto katote lithium waikawa valproic ranei ranei.

kawea Whakahohe te whakamahi o te whakararuraru, pourua i roto i te dosing rā tuatahi i roto i te 0.010 tūroro i whakamana ki te te fariiraa o te medicament mo mania whakapeka, kia tonu reira ki te whakamahi i te rauemi i roto i te taua moni.

disorders fakalotofo'í e pā ana ki te tūroro disorders pourua pakeke tukinotia ki te huinga o 0,005 go o olanzapine me 0,020 teuteu g fluoksetinovyh e e faaterehia i roto i te ahiahi.

pānga Antidepressive o te raau taero whakakitea i roto i te nui o i 0,006 ki te 0.012 karamu ki te dosing rā toharite i roto i 0,0074 g horopeta rongoa fluoksetinovyh pae i 0,025 ki te 0,030 g Ki te reira te mea he akiaki, he mea ka taea ki te whakahou i te dosing o raau taero e rua.

nekehia haumanu ahua pūmau o te korekore e te huinga o 0,005 g, me te 0.02 go o tikanga fluoksetinovyh olanzapine e whakahaerea nei kotahi i roto i te ahiahi.

Whakaahuatanga "Zyprexa" tarukino

Tenei neuroleptic whakaputaina i roto i te puka papa pani ki te takotoranga. E wha inenga waihanga: 0,0025 i 0,005, 0,010, me 0,0075 mo x, y e he momotuhi tika i runga i te mata «Lilly 4112», «Lilly 4115», «Lilly 4116», «Lilly 4117".

kai tautauā i roto i te puka o te reihuka, hydroxypropylcellulose, crospovidone, i hanga microcrystalline momo cellulose hanganga te o te konupora stearate rongoā.

Kua tākai nga papa i roto i te opupu o 7 nga wahi i roto i te mōkihi kei 4 aratau tākai.

He he ano hoki te puka Freeze-maroke, te tikanga mo te hanga o rongoā intramuscular. tākai Kōwhai 0.01g inenga wai ki oko. E whakaaro wāhanga hohekore monohydrate reihuka, me te waikawa tātariki.

whakaaturia te tarukino pānga ähotea.

Ko te whakauru mātātoa o te medicament e mahi rite ligand e herea ki te serotonin, dopamine, m-Matuorakouawai, H1-histamine me Alpha1-receptor ngā adrenozavisimymi. Olanzapine he pānga whiriwhiri i runga i te āhua o te pūnaha limbic.

Drug "Zyprexa" ako i runga i te tono tohutohu ki te whakamahi i ki ngā wāhanga kaha o disorders wairua tuakoi me psychotic e kua haere tahi e mārama tohu o horihori, moemoea, disorders whakaaro, kino, huru hihira ranei he momo kino i roto i te puka o te whakarerenga aronganui me te pāpori, disorders o te taputapu waiata. tohua te rongoā te mo te tango o nga tohu pängia Tuarua meinga e disorders wairua tuakoi.

Tablet "Zyprexa" ā-ako taunaki inu-waha, i tetahi wa. maimoatanga wawe o te horopeta kotahi ko te 0,010 g muri pae te inenga rā i 0,005 ki te 0,020 g, titia nei te ki pikitia symptomatic.

patia Intramuscularly rongoā, ki te ki he hiahia akiaki mutu te whakamātau tinana excitation pūāhua i roto i te iwi ki te wairua tuakoi, pourua disorders pängia me te tupu.

I mua i te whakamahi, diluted te lyophilisate i roto i 2.1 ml reo wai injectable. He otinga mārama ki te urukehu kōwhai.

Ko te oaoa manavasii o te whakararuraru, wairua tuakoi te, me te pourua tango atu i roto i te kotahi-horopeta o 0,010

Whakaaro inaianei te manawanui haumanu, whakamana whakahaere toutou o inenga 0,010 g i muri i 120 min i te tono tuatahi, me te 0,010 g e whai ake nei pau i muri i 240 meneti i te tono tuarua.

Hoki atu maimoatanga tarukino "Zyprexa" nekehanga ki tona puka papa ki te inenga o i 0,005 ki te 0,020 g

Ketia i roto i te dementia nekehia i roto i te horopeta intramuscular kotahi o 0,0025 Whakaaro te pikitia haumanu o te manawanui, kawea te rua o nga 0.005g whakahaere inenga i muri 120 meneti i te tono tuatahi.

whakaahuatanga Hua "Adair Zyprexa"

He medicament "olanzapine" analogs e kua whakaputaina i roto i te puka paura i 0,405 go o olanzapine i roto i te oko ki te pūwero whakarewa me te ngira.

Tikanga "Adair Zyprexa" e pā ana ki ähotea mahi taero neuroleptic.

Rongoā Kōpeke ino, kua whakamahia hoki te pupuri me te wā roa-maimoatanga o protivopovtornogo wairua tuakoi te me huringa hinengaro ki tohumate o tiketike-tukua i roto i te puka o horihori, i kitea hallucinatory me flattening kino aronganui, mauriora ki te taputapu waiata.

Medicines hamani nui wāhanga härukiruki me ngā o te whakararuraru, pourua, i roto i te mea e taea āhuatanga psychotic me te huringa tere i roto i ngā wāhanga.

whakamahia Initial inenga rā e 0.010 ranei 0.015, te nui o te tarukino tīpakohia mō ia manawanui takitahi rā, tango ki pūkete te pikitia haumanu. whakamahia Tikanga whakaora horopeta ia rā o i 0,005 ki te 0,020 g

Te whakanui ake i te inenga he taea anake ki nga hua o rangahau. Te whakanui ake i te nui o te tarukino kawea i roto i roto i ngā wāhanga, i nga ra.

tūroro kaumātua, te horopeta tuatahi rā i roto i te aroaro o te mahi tākihi iti me te ate tautapa 0.005 g

analogues utu

Whārangi nui o antipsychotics e āhei ki a koe te whiriwhiri i te tarukino tika, i te mea e tika ana i roto i te kounga me te utu. Rongoā "Olanzapine" he utu āhua iti. Ka taea te hokona Packaging o papa mo 290 moni.

Ko Drug "Zalasta" utu i 1370 moni.

whakaaro tikanga utu pire "Zidis Zyprexa." Hoki mōkihi hua Me ki utu 2370 moni. uara tairitenga o "Ku-Ripa Zalasta" Ko 1075 moni.

I rongoa riro "Zyprexa" utu arotake kino. He mōkihi o 28 papa utu 4760 moni.

No te rōpū rawakore e kia wātea tarukino "Olanzapine", i te mea he hautanga o te utu.

Tirohanga o tūroro

Mō ngā rongoā e taea te rongo "Olanzapine" arotake e rua pai, me te kino. tauturu tokomaha tarukino ki te akakoromaki i te whārua, me te whakaiti i te nui o whakaaro kino i muri i te torutoru nga ra o te maimoatanga. Kei te whakaaro ia tetahi o nga kaha o neuroleptics, e tamarû te manawanui, faaore wehi me manukanuka.

I roto i te āhuatanga emit pānga e hiahiatia e e pā ana ki te tērā o te pākia, hua i roto i nui haere taimaha o te manawanui tinana. Somnolence, asthenia syndrome, whanoke, kia maturuturu toto orthostatic momo pēhanga whakawhanake kiko ngohengohe puku me te maroke o kiriuhi mucous.

No te tahi mau tūroro, ara he horopeta iti o te rongoā ko te whakarokiroki kaha, i nei moe ratou mo 12 haora i te ra.

Ko te tinana tangata rerekē, Heoi, ka whakahihi rerekē papa mo ia manawanui. Me hoki te kōwhiringa o taputapu e tika ana ki te kōrero i te tākuta.

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